A proposed inhalation reference concentration for methanol

Starr, TB; Festa, JL

HERO ID

52598

Reference Type

Journal Article

Subtype

Review

Year

2003

Language

English

PMID

14550762

HERO ID 52598
Material Type Review
In Press No
Year 2003
Title A proposed inhalation reference concentration for methanol
Authors Starr, TB; Festa, JL
Journal Regulatory Toxicology and Pharmacology
Volume 38
Issue 2
Page Numbers 224-231
Abstract A biologically based approach was taken to developing an inhalation Reference Concentration (RfC) for methanol, a high production volume chemical with many commercial applications, including use as an alternative fuel for motor vehicles and as a hydrogen source for fuel cells. Benchmark Dose methodology was applied to the most sensitive toxic endpoint for assessing potential health risks in humans, cervical rib malformation data obtained using CD-1 mice. The concentration of methanol in circulating blood was employed as the dose metric, and the maximum likelihood estimate of the blood methanol increment causing a 10% extra risk of these malformations, was 215.4 mg/L, with a lower 95% confidence bound of 97.4 mg/L. A "Reference Increment" for blood methanol was then determined by dividing this value by a 3-fold factor for residual pharmacodynamic uncertainty between species and a 10-fold factor for interindividual variation in human sensitivity to methanol. The resulting Reference Increment in blood methanol was then converted to an equivalent inhalation Reference Concentration with a physiologically based pharmacokinetic model evaluated for continuous exposure conditions. The resulting maximum likelihood estimate for the inhalation RfC was 298 mg/m3, with a 95% lower confidence bound of 135 mg/m3.
Pmid 14550762
Wosid WOS:000186079800010
Is Certified Translation No
Dupe Override No
Comments ECRIB.Regul. Toxicol. Pharmacol. 38: 224-231.
Is Public Yes
Language Text English
Keyword Abnormalities, Drug-Induced/etiology; Administration, Inhalation; Animals; Environmental Pollutants/administration & dosage/pharmacokinetics/toxicity; Female; Humans; Maternal-Fetal Exchange; Methanol/administration & dosage/pharmacokinetics/toxicity; Mice; Models, Animal; Pregnancy; Reference Values; Risk Assessment; Species Specificity; 0 (Environmental Pollutants); 67-56-1 (Methanol)
Is Qa No