The acidity and self-catalyzed lactonization of l-gulonic acid: Thermodynamic, kinetic and computational study

Kutus, B; Peintler, G; Buckó, Á; Balla, Z; Lupan, A; Attia, AAA; Pálinkó, I; Sipos, P

HERO ID

4943165

Reference Type

Journal Article

Year

2018

Language

English

PMID

30048821

HERO ID 4943165
In Press No
Year 2018
Title The acidity and self-catalyzed lactonization of l-gulonic acid: Thermodynamic, kinetic and computational study
Authors Kutus, B; Peintler, G; Buckó, Á; Balla, Z; Lupan, A; Attia, AAA; Pálinkó, I; Sipos, P
Journal Carbohydrate Research
Volume 467
Page Numbers 14-22
Abstract Lactonization and proton dissociation of sugar acids take place simultaneously in acidic aqueous solutions. The protonation-deprotonation processes are always fast, whilst the formation and hydrolysis of γ- and δ-lactones are usually slower. Thus, both thermodynamic and kinetic information are required for the complete understanding of these reactions. The protonation constant (Kp) of l-gulonate (Gul-) was determined from potentiometric and polarimetric measurements, while the individual lactonization constants (KL,γ and KL,δ) for l-gulonic acid (HGul) were obtained via13C NMR experiments. The applicability of this method was proven by measuring these well-known constants for d-gluconic acid (HGluc) and by comparing them to literature data. l-gulonic acid γ-lactone (γ-HGul) has remarkable stability in contrast with δ-HGul as well as γ- and δ-HGluc. The polarimetric measurement implies that the main factor responsible for the enhanced stability of γ-HGul is that its hydrolysis is much slower than that of δ-HGul. This higher stability of the γ-HGul ring over its δ-isomer was also confirmed by quantum chemical calculations. A new confirmed feature of the reaction is that in parallel to H3O+, HGul also catalyzes the formation and reverse hydrolytic processes of γ-HGul, similarly to other general acid catalysts.
Doi 10.1016/j.carres.2018.07.006
Pmid 30048821
Wosid WOS:000441886200003
Is Certified Translation No
Dupe Override No
Is Public Yes
Language Text English