Rapid preparation of (methyl)malonyl coenzyme A and enzymatic formation of unusual polyketides by type III polyketide synthase from Aquilaria sinensis

Gao, BW; Wang, XH; Liu, X; Shi, SP; Tu, PF

HERO ID

3537907

Reference Type

Journal Article

Year

2015

Language

English

PMID

25677661

HERO ID 3537907
In Press No
Year 2015
Title Rapid preparation of (methyl)malonyl coenzyme A and enzymatic formation of unusual polyketides by type III polyketide synthase from Aquilaria sinensis
Authors Gao, BW; Wang, XH; Liu, X; Shi, SP; Tu, PF
Journal Bioorganic & Medicinal Chemistry Letters
Volume 25
Issue 6
Page Numbers 1279-1283
Abstract (Methyl)malonyl coenzyme A was rapidly and effectively synthesized by a two-step procedure involving preparation of N-hydroxysuccinimidyl (methyl)malonate from (methyl)Meldrum's acid, and followed by transesterification with coenzyme A. The synthesized (methyl)malonyl coenzyme A could be well accepted and assembled to 4-hydroxy phenylpropionyl coenzyme A by type III polyketide synthase from Aquilaria sinensis to produce dihydrochalcone and 4-hydroxy-3,5-dimethyl-6-(4-hydroxyphenethyl)-2H-pyrone as well as 4-hydroxy-3,5-dimethyl-6-(5-(4-hydroxyphenyl)-3-oxopentan-2-yl)-2H-pyrone.
Doi 10.1016/j.bmcl.2015.01.045
Pmid 25677661
Wosid WOS:000350696000022
Is Certified Translation No
Dupe Override No
Comments Journal: Bioorganic & medicinal chemistry letters ISSN: 1464-3405
Is Public Yes
Language Text English