Enhancement of Thioredoxin Production from Nasal Epithelial Cells by the Macrolide Antibiotic, Clarithromycin In Vitro

Suzaki, I; Asano, K; Kanei, A; Suzaki, H

HERO ID

2289214

Reference Type

Journal Article

Year

2013

PMID

23606690

HERO ID 2289214
In Press No
Year 2013
Title Enhancement of Thioredoxin Production from Nasal Epithelial Cells by the Macrolide Antibiotic, Clarithromycin In Vitro
Authors Suzaki, I; Asano, K; Kanei, A; Suzaki, H
Journal In Vivo
Volume 27
Issue 3
Page Numbers 351-356
Abstract Low-dose and long-term administration of 14-membered macrolide antibiotics is well-known to be effective in the treatment of chronic airway diseases. Although there is much evidence that the anti-inflammatory action, but not the anti-microbial action of macrolides, is responsible for the clinical efficacy of these agents on chronic airway inflammatory diseases, the precise therapeutic mechanisms are not well-understood. Since thioredoxin (TRX) has now attracted attention as an endogenous peptide with immunomodulatory effects, the present study was undertaken to examine whether macrolide antibiotics could favorably modulate the clinical status of such diseases via the production of TRX from nasal epithelial cells in vitro. Nasal epithelial cells (5x10(5) cells/ml) obtained from five patients were stimulated with 50 mu M H2O2 in the presence of different concentrations of macrolide antibiotics for 24 h. TRX levels in culture supernatants were examined by enzyme-linked immunosorbent assay. We also examined the influence of macrolide antibiotics on TRX mRNA expression and mRNA translation by RT-PCR and a wheat germ cell-free protein synthesis technique, respectively. The addition of clarithromycin (CAM) to cell cultures caused an increase in the ability of cells to produce TRX in response to H2O2 stimulation, and the minimum concentration that caused a significant increase was 0.5 mu g/ml. On the other hand, josamycin, a 16-membered macrolide antibiotic, did not increase TRX production induced by H2O2 stimulation. Although the treatment of cells with CAM inhibits TRX mRNA transcription, the agent might increase translation of mRNA to produce specific proteins. The ability of CAM to increase TRX production may account, at least in part, for the clinical efficacy of this agent on chronic airway inflammatory diseases, including chronic rhinosinositis.
Pmid 23606690
Wosid WOS:000318319100008
Is Certified Translation No
Dupe Override No
Is Public Yes
Keyword Thioredoxin; clarithromycin; chronic airway inflammatory diseases; nasal epithelial cells