Acute effects of polychlorinated biphenyl-containing and -free transformer fluids on rat testicular steroidogenesis

Andric, SA; Kostic, TS; Dragisic, SM; Andric, NL; Stojilkovic, SS; Kovacevic, RZ

HERO ID

1415639

Reference Type

Journal Article

Year

2000

Language

English

PMID

11049815

HERO ID 1415639
In Press No
Year 2000
Title Acute effects of polychlorinated biphenyl-containing and -free transformer fluids on rat testicular steroidogenesis
Authors Andric, SA; Kostic, TS; Dragisic, SM; Andric, NL; Stojilkovic, SS; Kovacevic, RZ
Journal Environmental Health Perspectives
Volume 108
Issue 10
Page Numbers 955-959
Abstract Polychlorinated biphenyl (PCB)-based transformer fluids belong to a class of environmentally persistent mixtures with known toxic effects. Here, we studied the acute effects of Askarel (which contains Aroclor 1260) and two substitute transformer fluids (the silicone oil-based DC561 and the mineral oil-based ENOL C) on rat testicular steroidogenesis. Single intraperitoneal (ip; 10 mg/kg body weight) or bilateral intratesticular (itt; 25 microg/testis) injections of Askarel markedly decreased serum androgen levels 24 hr after administration. In acute testicular cultures from these animals, chorionic gonadotropin-stimulated progesterone and androgen productions were severely attenuated. When itt was injected or added in vitro, Askarel inhibited 3ss-hydroxysteroid dehydrogenase (3ssHSD), stimulated 17[alpha]-hydroxylase/lyase (P450c17), and did not affect 17ss-hydroxysteroid dehydrogenase in testicular postmitochondrial fractions. The ip-injected Askarel did not affect 3ssHSD, but inhibited P450c17, suggesting that a more intensive metabolism of peripherally injected Askarel reduces the circulating levels of active ingredients below the threshold needed for inhibition of 3ssHSD and generates a derivative that inhibits P450c17. In contrast to Askarel, itt-injection (25 microg/testis) of DC561 and ENOL C did not affect in vivo and in vitro steroidogenesis. These findings show the acute effects of Askarel, but not silicone and mineral oils, on testicular steroidogenesis.
Doi 10.1289/ehp.00108955
Pmid 11049815
Wosid WOS:000090093000022
Is Certified Translation No
Dupe Override No
Is Public Yes
Language Text English
Keyword 3 beta-hydroxysteroid dehydrogenase; androgen; P450c17; polychlorinated biphenyls; progesterone
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