Diastereoselectivity of additions to chiral carbonyl oxides

Dussault, PH; Zope, UR

HERO ID

1193209

Reference Type

Journal Article

Year

1995

HERO ID 1193209
In Press No
Year 1995
Title Diastereoselectivity of additions to chiral carbonyl oxides
Authors Dussault, PH; Zope, UR
Journal Journal of Organic Chemistry
Volume 60
Issue 25
Page Numbers 8218-8222
Abstract The influence of a resident stereocenter on the formation of hydroperoxy acetals from carbonyl oxides is investigated. Addition of either methanol or 2-propanol to 8-phenylpropanal O-oxide proceeds with modest stereoselectivity; addition of a tertiary alcohol proceeds with higher selectivity. Product stereochemistry, which is confirmed by conversion of a functionalized hydroperoxy acetal to a 1,2-dioxane, is found to derive from nucleophilic attack through a Felkin-Anh type transition state. Trapping of a carbonyl oxide containing a neighboring hydrogen bond donor proceeds with modest selectivity for both syn- and anti-carbonyl oxide isomers. Ozonolysis of a 3-(trialkylstannyl)-1-enol ether proceeds with loss of the stannyl-bearing carbon through the possible intermediacy of a vinyl peroxide.<
Doi 10.1021/jo00130a021
Wosid WOS:A1995TK91900021
Is Certified Translation No
Dupe Override No
Comments Source: Web of Science A1995TK91900021
Is Public Yes
Is Qa No